bx - 528 |
目标 |
羧肽酶B |
细节 |
(2 s) - n - [(3 e) 5-cyclopropyl-3h-pyrazol-3-ylidene] 2 - [4 - (2-oxo-1-imidazolidinyl)苯基]丙酰胺 |
目标 |
细胞周期蛋白依赖性激酶2 |
细节 |
(2 s) - n - [(3 e) 5-cyclopropyl-3h-pyrazol-3-ylidene] 2 - [4 - (2-oxo-1-imidazolidinyl)苯基]丙酰胺 |
目标 |
Cyclin-A2 |
细节 |
Neflamapimod |
目标 |
增殖蛋白激酶14 |
细节 |
3 - (5 - (3-nitrophenyl) thiophen-2-yl]丙酸 |
目标 |
醛糖还原酶 |
细节 |
5 - [(3 r) 3 - (5-methoxybiphenyl-3-yl) but-1-yn-1-yl] 6-methylpyrimidine-2, 4-diamine |
目标 |
二氢叶酸还原酶 |
细节 |
5 - [(3 r) 3 - (5-methoxybiphenyl-3-yl) but-1-yn-1-yl] 6-methylpyrimidine-2, 4-diamine |
目标 |
二氢叶酸还原酶(dfrB) |
细节 |
5 - [(3 r) 3 - (5-methoxy-4 -methylbiphenyl-3-yl) but-1-yn-1-yl] 6-methylpyrimidine-2 4-diamine |
目标 |
二氢叶酸还原酶 |
细节 |
5 - [3 - (3 r) (5-methoxy-3 ', 5 ' -dimethylbiphenyl-3-yl) but-1-yn-1-yl] 6-methylpyrimidine-2, 4-diamine |
目标 |
二氢叶酸还原酶(dfrB) |
细节 |
5 - [3 - (3 r) (5-methoxy-3 ', 5 ' -dimethylbiphenyl-3-yl) but-1-yn-1-yl] 6-methylpyrimidine-2, 4-diamine |
目标 |
二氢叶酸还原酶 |
细节 |
D-phenylalanyl-N-benzyl-L-prolinamide |
目标 |
凝血酶原 |
细节 |
5 - [3 - (3 r) (5-methoxy-2 ', 6 ' -dimethylbiphenyl-3-yl) but-1-yn-1-yl] 6-methylpyrimidine-2, 4-diamine |
目标 |
二氢叶酸还原酶 |
细节 |
(2 r) -N-HYDROXY-2 - [(3 s) 3-methyl-3 - {4 - [(2-METHYLQUINOLIN-4-YL)甲氧基]苯基}2-oxopyrrolidin-1-yl]丙酰胺 |
目标 |
Disintegrin和金属蛋白酶domain-containing蛋白17 |
细节 |
(2,3-DIPHENYL-N) - 2-PIPERAZIN-1-YLETHYL FURO [2, 3 b] PYRIDIN-4-AMINE |
目标 |
酪氨酸受体激酶Lck |
细节 |
甲基(1 r, 2 s) 2 - (hydroxycarbamoyl) 1 - {4 - [(2-methylquinolin-4-yl)甲氧基]苄}cyclopropanecarboxylate |
目标 |
Disintegrin和金属蛋白酶domain-containing蛋白17 |
细节 |
(6 s) 1-chloro-3 - [(4-fluorobenzyl)氧]6 - (pyrrolidin-1-ylcarbonyl) pyrrolo (1 a) pyrazin-4——(6小时) |
目标 |
Prolyl肽链内切酶 |
细节 |
(7)2 - (2-aminopyrimidin-4-yl) 7 - (2-fluoroethyl) 1、5、6, 7-tetrahydro-4H-pyrrolo [3、2 c] pyridin-4-one |
目标 |
糖原合成酶激酶3β |
细节 |
(4)- 4-HYDROXYPHENYL 1-naphthaldehyde肟 |
目标 |
雌激素受体β |
细节 |
(4)- 4-HYDROXYPHENYL 1-naphthaldehyde肟 |
目标 |
核受体共激活剂1 |
细节 |
(4)- 4-hydroxy-3-methylphenyl 6-phenylpyrimidin-2——(5小时) |
目标 |
丝氨酸/ threonine-protein激酶pim-1 |
细节 |
N - (4 - (5-fluoro-6-methylpyridin-2-yl) 5-quinoxalin-6-yl-1h-imidazol-2-yl)乙酰胺 |
目标 |
鉴定及受体1型 |
细节 |
6-methyl-5 - [3-methyl-3 (3、4、5-trimethoxyphenyl) but-1-yn-1-yl] pyrimidine-2, 4-diamine |
目标 |
二氢叶酸还原酶(dfrB) |
细节 |
(3 r) 4 - [(3 r) 3-amino-4 - (2, 4, 5-TRIFLUOROPHENYL) BUTANOYL] 3-methyl-1, 4-DIAZEPAN-2-ONE |
目标 |
Dipeptidyl肽酶4 |
细节 |
(3 s) 1-cyclohexyl-5-oxo-n-phenylpyrrolidine-3-carboxamide |
目标 |
Enoyl——(酰基载体蛋白质)还原酶(NADH) |
细节 |
(4 z) 6-bromo-4 ({[4 - (pyrrolidin-1-ylmethyl)苯基]氨基}methylidene) isoquinoline-1, 3 (2 h, 4 h)土卫四 |
目标 |
胰岛素样生长因子1受体 |
细节 |
(5 r, 6、8) 8 -[3 -(氨甲基)苯基]6-hydroxy-5-isopropyl-3-oxo-1-phenyl-2 7-DIOXA-4-AZA-6-PHOSPHANONAN-9-OIC酸6-OXIDE |
目标 |
羧肽酶B |
细节 |
5-ETHYL-3-METHYL-1, 5-DIHYDRO-4H-PYRAZOLO [4、3 c] QUINOLIN-4-ONE |
目标 |
丝氨酸/ threonine-protein激酶Chk1 |
细节 |
Tamatinib |
目标 |
酪氨酸受体激酶麦克米兰 |
细节 |
N - {((2 s, 3 s) 3 -(乙氧羰基)OXIRAN-2-YL]羰基}-L-ISOLEUCINE |
目标 |
组织蛋白酶B |
细节 |
5-phenyl-1H-indazol-3-amine |
目标 |
酪氨酸受体激酶JAK2 |
细节 |