Serotonin 4 Receptor Agonists
- Name
- Serotonin 4 Receptor Agonists
- Accession Number
- DBCAT005477
- Description
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Not Available
- Drugs
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Drug Drug Description Prucalopride A 5-HT4 receptor agonist indicated to treat adults with chronic idiopathic constipation. Tegaserod A serotonin-4 (5-HT4) receptor agonist indicated for the treatment of constipation predominant irritable bowel syndrome (IBS-C) specifically in women under the age of 65. There is currently no safety or efficacy data for use of tegaserol in men. - Drugs & Drug Targets
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Drug Target Type Prucalopride 5-hydroxytryptamine receptor 4 target Prucalopride Cytochrome P450 3A4 enzyme Prucalopride Serum albumin carrier Prucalopride P-glycoprotein 1 transporter Tegaserod 5-hydroxytryptamine receptor 4 target Tegaserod 5-hydroxytryptamine receptor 2B target Tegaserod 5-hydroxytryptamine receptor 2C target Tegaserod 5-hydroxytryptamine receptor 2A target Tegaserod Sodium-dependent serotonin transporter transporter Tegaserod Cytochrome P450 1A2 enzyme Tegaserod Cytochrome P450 2C8 enzyme Tegaserod Cytochrome P450 2D6 enzyme Tegaserod Cytochrome P450 2E1 enzyme Tegaserod ATP-binding cassette sub-family G member 2 transporter Tegaserod P-glycoprotein 1 transporter