Serotonin 1b Receptor Agonists

Name
Serotonin 1b Receptor Agonists
Accession Number
DBCAT004121
Description

Not Available

Drugs
Drug Drug Description
Almotriptan A 5-HT1B/1D receptor agonist used to treat migraines.
Zolmitriptan A member of the triptan class of 5-HT(1B/1D/1F) receptor agonist drugs used for the acute treatment of migraine with or without aura in adults.
Sumatriptan A serotonin receptor agonist used to treat migraines and cluster headaches.
Naratriptan A 5-HT1B/1D receptor agonist used to treat migraines.
Rizatriptan A 5-HT1B/1D receptor agonist used to treat migraines.
Frovatriptan A 5-HT1B/1D receptor agonist used to treat migraines.
Eletriptan A triptan used for the treatment of migraines.
Drugs & Drug Targets
Drug Target Type
Almotriptan 5-hydroxytryptamine receptor 1D target
Almotriptan 5-hydroxytryptamine receptor 1B target
Almotriptan Cytochrome P450 3A4 enzyme
Almotriptan Cytochrome P450 2D6 enzyme
Almotriptan Amine oxidase [flavin-containing] A enzyme
Almotriptan Dimethylaniline monooxygenase [N-oxide-forming] 3 enzyme
Almotriptan Cytochrome P450 2C19 enzyme
Almotriptan Cytochrome P450 2E1 enzyme
Almotriptan Cytochrome P450 2C8 enzyme
Zolmitriptan 5-hydroxytryptamine receptor 1D target
Zolmitriptan 5-hydroxytryptamine receptor 1B target
Zolmitriptan 5-hydroxytryptamine receptor 1F target
Zolmitriptan Cytochrome P450 1A2 enzyme
Zolmitriptan Amine oxidase [flavin-containing] A enzyme
Zolmitriptan 5-hydroxytryptamine receptor 1A target
Zolmitriptan P-glycoprotein 1 transporter
Zolmitriptan 5-hydroxytryptamine receptor 7 target
Zolmitriptan 5-hydroxytryptamine receptor 2A target
Zolmitriptan 5-hydroxytryptamine receptor 2B target
Zolmitriptan 5-hydroxytryptamine receptor 1E target
Sumatriptan 5-hydroxytryptamine receptor 1D target
Sumatriptan 5-hydroxytryptamine receptor 1B target
Sumatriptan 5-hydroxytryptamine receptor 1F target
Sumatriptan Amine oxidase [flavin-containing] A enzyme
Sumatriptan 5-hydroxytryptamine receptor 1A target
Sumatriptan Solute carrier organic anion transporter family member 1A2 transporter
Sumatriptan P-glycoprotein 1 transporter
Sumatriptan ATP-binding cassette sub-family G member 2 transporter
Sumatriptan Solute carrier organic anion transporter family member 1B1 transporter
Naratriptan 5-hydroxytryptamine receptor 1D target
Naratriptan 5-hydroxytryptamine receptor 1B target
Naratriptan 5-hydroxytryptamine receptor 1F target
Naratriptan 5-hydroxytryptamine receptor 1A target
Naratriptan Amine oxidase [flavin-containing] A enzyme
Rizatriptan 5-hydroxytryptamine receptor 1D target
Rizatriptan 5-hydroxytryptamine receptor 1B target
Rizatriptan 5-hydroxytryptamine receptor 1F target
Rizatriptan Amine oxidase [flavin-containing] A enzyme
Frovatriptan 5-hydroxytryptamine receptor 1D target
Frovatriptan 5-hydroxytryptamine receptor 1B target
Frovatriptan Cytochrome P450 1A2 enzyme
Eletriptan 5-hydroxytryptamine receptor 1D target
Eletriptan 5-hydroxytryptamine receptor 1A target
Eletriptan 5-hydroxytryptamine receptor 1F target
Eletriptan 5-hydroxytryptamine receptor 1B target
Eletriptan Cytochrome P450 3A4 enzyme
Eletriptan Cytochrome P450 2D6 enzyme
Eletriptan Cytochrome P450 2C9 enzyme
Eletriptan Cytochrome P450 2C19 enzyme
Eletriptan Prostaglandin G/H synthase 1 enzyme
Eletriptan Cytochrome P450 2A6 enzyme
Eletriptan P-glycoprotein 1 transporter